PMID: 42213035

Discovery of an Androgen Receptor Degrader Featuring a Pyridazinyl Glutarimide CRBN-Binding Motif for Transdermal Treatment of Androgenetic Alopecia.

Wang Xiao, Ge Ling, Yu Yawei, Zhong Tengjiang, Hu Weitong, Zhang Sai, Chen Xuan, Yang Miaoyuan, Zhang Xinxin, Li Zhuoyue

Journal of medicinal chemistry · 2026

Vol. 69, Issue 11, pp. 13028-13054

This entry links to third-party literature. For research use only.

AnimalsAlopeciaReceptors, AndrogenHumansMiceProteolysis Targeting ChimeraMaleUbiquitin-Protein LigasesAdministration, CutaneousPyridazines

For research use only. This index links to third-party literature. Nothing here constitutes medical advice.