PMID: 42213035
Discovery of an Androgen Receptor Degrader Featuring a Pyridazinyl Glutarimide CRBN-Binding Motif for Transdermal Treatment of Androgenetic Alopecia.
Wang Xiao, Ge Ling, Yu Yawei, Zhong Tengjiang, Hu Weitong, Zhang Sai, Chen Xuan, Yang Miaoyuan, Zhang Xinxin, Li Zhuoyue
Journal of medicinal chemistry · 2026
Vol. 69, Issue 11, pp. 13028-13054
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AnimalsAlopeciaReceptors, AndrogenHumansMiceProteolysis Targeting ChimeraMaleUbiquitin-Protein LigasesAdministration, CutaneousPyridazines